Programme
TUESDAY 21ST FEBRUARY 2017 |
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13:15 – 14:15 |
Registration & Reception |
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13:15 – 14:15 |
Welcome Lunch |
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14:15 – 14:30 |
Opening Comments |
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NEW APPROACHES IN BIOTECH AND ACADEMIA |
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14:30 – 15:15 |
Ted Torphy |
“IN THEORY, THE MODEL IS BRILLIANT” – LEARNINGS FROM THE HARRINGTON PROJECT, A NEW DISTRIBUTIVE MODEL OF R&D |
15:15 – 15:45 |
Guy Breitenbucher |
REFLECTING ON FATTY ACID AMIDE HYDROLASE (FAAH): A LOOK BACK AT A SUCCESSFUL ACADEMIC-INDUSTRIAL COLLABORATION IN DRUG DISCOVERY |
15:45 – 16:15 |
Bob Wenslow |
DON’T OVERLOOK KEY PRECLINICAL RESEARCH IN EARLY PHARMACEUTICAL DEVELOPMENT |
16:15 – 16:45 |
Refreshments |
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NEW APPROACHES IN BIOTECH AND ACADEMIA |
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16:45 – 17:15 |
Kevin Madauss |
GSK’s TRUST IN SCIENCE PROGRAM: AN ALTERNATIVE DISCOVERY AND DEVELOPMENT MODEL IN LATIN AMERICA |
17:15 – 17:45 |
Jose Fernandez |
FROM CONSUMER PRODUCTS TO DRUGS: DEVELOPING NOVEL TECHNOLOGIES IN DERMATOLOGY AND NEUROLOGY |
17:45 – 18:15 |
Garry Smith |
DRUG DISCOVERY AT THE ACADEMIC/BIOTECH START-UP INTERFACE: DEVELOPMENT OF SMALL MOLECULES TO TREAT EPSTEIN-BARR VIRUS-ASSOCIATED DISEASES, CONTINUED |
18:15 – 18:45 |
Stephen Martin |
APPLICATIONS OF CHEMISTRY TO UNMET MEDICAL NEEDS IN NEUROSCIENCE |
18:45 |
Dinner at Leisure & Free Time |
WEDNESDAY 22ND FEBRUARY 2017 |
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07:00 – 08:15 |
Breakfast *Kalmia Buffet Restaurant* |
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NATURAL PRODUCTS SESSION |
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08:15 – 08:30 |
Cedric Pearce |
INTRODUCTORY COMMENTS |
08:30 – 09:15 |
Nicholas Oberlies |
ANTICANCER DRUG LEADS FROM NATURAL SOURCES: STRATEGIES, PROGRESS, AND INNOVATIVE TECHNIQUES |
09:15 – 09:45 |
Roberto Berlinck |
DISCOVERY AND SAR INVESTIGATIONS OF ANTI-PARASITIC ALKALOIDS |
09:45 – 10:15 |
Jose Medina |
CHEMINFORMATICS ANALYSIS OF THE CHEMICAL SPACE OF NATURAL PRODUCTS FOR DRUG DISCOVERY |
10:15 – 10:45 |
Refreshments & Group Photo |
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10:45 – 11:15 |
Guy Carter |
LEVERAGING THE CHEMICAL DIVERSITY OF AQUATIC MICROBIOMES |
11:15 – 11:45 |
Mark Hamann |
NUISANCE AND HARMFUL ALGAL BLOOMS: AN EMERGING SOURCE FOR DRUG DISCOVERY AND DEVELOPMENT |
11:45 –12:15 |
Ronald Quinn |
FRAGMENT-BASED DRUG DISCOVERY USING NATURAL PRODUCTS |
12:15 –12:45 |
Andreas Vilcinskas |
THE SANOFI-FRAUNHOFER CENTER FOR NAURAL PRODUCT RESEARCH |
12:45 – 16:15 |
Lunch at Leisure & Free Time |
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NON-PROFIT SECTOR IN DRUG DISCOVERY AND DEVELOPMENT |
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16:15 – 16:45 |
Peter Warner |
DRUG DISCOVERY FOR NEGLECTED DISEASES: IMPORTANCE OF PARTNERSHIPS |
16:45 – 17:15 |
Leah Frye |
STRUCTURE-BASED DRUG DISCOVERY IN THE NON-PROFIT SECTOR |
17:15 – 17:45 |
Jeremy Burrows |
DRUG DISCOVERY TO CONTROL AND ERADICATE MALARIA |
17:45 – 18:15 |
Refreshments |
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18:15 – 18:45 |
Manu De Rycker |
DISCOVERY AND LEAD-OPTIMISATION OF A PROMISING NEW ANTILEISHMANIAL COMPOUND SERIES WITHIN AN ACADEMIC-INDUSTRY PARTNERSHIP |
18:45 – 19:15 |
Barry Bunin |
PRESENT AND FUTURE COLLABORATIVE DRUG DISCOVERY INFORMATICS INNOVATIONS |
19:15 – 19:45 |
Christopher B. Cooper |
ANTITUBERCULAR 3-(4-AMINOPHENYL)OXAZOLIDIN-2-ONES: PROGRESS TOWARDS BETTER, SAFER TB AGENTS |
19:45 |
Dinner at Leisure & Free Time |
THURSDAY 23RD FEBRUARY 2017 |
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07:00 – 08:30 |
Breakfast *Kalmia Buffet Restaurant* |
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STRUCTURE, MODELING, AND FRAGMENT-BASED DESIGN SESSION |
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08:30 – 09:00 |
Dagmar Ringe |
CHEMICAL CHAPERONES AS AN APPROACH TO TREAMENT OF ALZHEIMER’S DISEASE |
09:00 – 09:30 |
Bill Jorgensen |
COMPUTER-AIDED DISCOVERY OF ENZYME INHIBITORS |
09:30 – 10:00 |
John Kulp |
AN OPEN WEB SERVICE FOR FRAGMENT-BASED DESIGN OF SMALL MOLECULES |
10:00 – 10:30 |
Refreshments |
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10:30 – 11:00 |
Chuck Reynolds |
RETHINKING LIGAND EFFICIENCY |
11:00 – 11:30 |
Matt Segall |
SEAMLESS INTEGRATION OF 3D STRUCTURE-BASED DESIGN AND 2D STRUCTURE-ACTIVITY RELATIONSHIPS TO GUIDE MEDICINAL CHEMISTRY |
11:30 – 12:00 |
Sandor Vajda |
HOT SPOT ANALYSIS FOR DRUGGABILITY AND FRAGMENT BINDING |
12:00 – 16:00 |
Lunch at Leisure & Free Time |
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DRUG DISCOVERY AND DEVELOPMENT TOOLS AND TECHNOLOGIES Session Chair: Bill Kinney, IteraMed Consulting |
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16:00 – 16:30 |
Rachel Garlish |
NATIVE AND HYDROGEN DEUTERIUM MASS SPECTROMETRY IN DRUG DISCOVERY |
16:30 – 17:00 |
Andrea L.C. Reid |
FOUNDATIONS OF PATENT LAW: OBVIOUSNESS |
17:00 – 17:30 |
Janet Ralbovsky |
DRUG DISCOVERY AND COMMERCIALIZATION AT THE DANA-FARBER CANCER INSTITUTE |
17:30 – 17:50 |
Martina Sutovska |
ECHINACEA PURPUREA - A SOURCE OF GLYCOCONJUGATE WITH BRONCHODILATING AND ANTI-INFLAMMATORY EFFECTS |
17:50 – 19:00 |
Poster Session & Refreshments |
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17:50 – 19:00 |
Andrea Reid (Dechert LLP) IP Breakout Session |
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19:30 |
*Gala Dinner & Poster Awards* |
FRIDAY 24TH FEBRUARY 2017 |
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07:00 – 08:30 |
Breakfast *Kalmia Buffet Restaurant* |
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NON-TRADITIONAL TARGETS AND APPROACHES |
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08:30 – 09:00 |
Scott Dax |
PHENOTYPIC SCREENING AND ANTI-OXIDANT ASSAYS LEADING TO THE DISCOVERY OF A NOVEL CLASS OF ANALGESICS |
09:00 – 09:30 |
Bart DeCorte |
NATURAL-PRODUCT DERIVED NOVEL CHEMICAL SPACE – A POWERFUL STARTING POINT IN DRUG DISCOVERY |
STUDENT PRESENTATIONS |
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09:30 – 09:50 |
Chao Wang |
MEET THE CHALLENGE: PROBING PARKINSON’S DISEASE BIOLOGY BY INTEGRATED MULTIDISCIPLINARY METHODOLOGY
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09:50 – 10:10 |
Xioayan Chen |
EXPLORATION OF DRUG LEADS FROM THE HUMAN MICROBIOME: AKKERMANSIA MUCINIPHILA |
10:10 – 10:25 |
Closing Comments |